Search results for "Biopartitioning micellar chromatography"

showing 2 items of 2 documents

Biopartitioning micellar chromatography to pedict mutagenicity of aromatic amines

2007

[EN] Mutagenicity is a toxicity endpoint associated with the chronic exposure to chemicals. Aromatic amines have considerable industrial and environmental importance due to their widespread use in industry and their mutagenic capacity. Biopartitioning micellar chromatography (BMC), a mode of micellar liquid chromatography that uses micellar mobile phases of Brij35 in adequate experimental conditions, has demonstrated to be useful in mimicking the drug partitioning process into biological systems. In this paper, the usefulness of BMC for predicting mutagenicity of aromatic amines is demonstrated. A multiple linear regression (MLR) model based on BMC retention data is proposed and compared wi…

Chronic exposureQuantitative structure–activity relationshipPredictive capabilityQuantitative Structure-Activity RelationshipAromatic aminesHigh-performance liquid chromatographyModels BiologicalMutagenicityDrug DiscoveryQUIMICA ANALITICAOrganic chemistryComputer SimulationAminesLeast-Squares AnalysisMicellesPharmacologychemistry.chemical_classificationChromatographyChromatographyOrganic ChemistryAromatic amineGeneral MedicineBiopartitioning micellar chromatographychemistryMicellar liquid chromatographyMutagenesisQuantitative retentione-activity relationships
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Biopartitioning micellar chromatoraphy to predict blood to lung, blood to liver, blood to fat and blood to skin partition coefficients of drugs

2009

[EN] Biopartitioning micellar chromatography (BMC), a mode of micellar liquid chromatography that uses micellar mobile phases of Brij35 in adequate experimental conditions, has demonstrated to be useful in mimicking the drug partitioning process into biological systems. In this paper, the usefulness of BMC for predicting the partition coefficients from blood to lung, blood to liver. blood to fat and blood to skin is demonstrated. PLS2 and multiple linear regression (MLR) models based on BMC retention data are proposed and compared with other ones reported in bibliography. The proposed models present better or similar descriptive and predictive capability. (C) 2008 Elsevier B.V. All rights r…

Quantitative structure–activity relationshipBlood to skinQuantitative Structure-Activity RelationshipPredictive capabilityPartition coefficientsBiochemistryAnalytical ChemistryPharmacokineticsBlood to lungLinear regressionQUIMICA ANALITICAmedicineAnimalsHumansEnvironmental ChemistryPharmacokineticsTissue DistributionLungMicellesSpectroscopySkinLungChromatographyChemistryComputational BiologyChromatography liquidBiopartitioning micellar chromatographyRatsPartition coefficientmedicine.anatomical_structureAdipose TissueLiverPharmaceutical PreparationsMicellar liquid chromatographyLinear ModelsBlood to fatRabbitsChromatography LiquidBlood to liver
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